Antidepressant & Psychedelic Drug Interaction Chart

Disclaimer: This chart is for informational purposes only and should not be used to make medical decisions. It is based on available data and some extrapolation. Decisions to start, stop, or taper medication and/or use psychedelic substances should always be made in consultation with your healthcare provider(s). Engaging in illicit activities is not recommended. For personal use only; do not copy or distribute.

Key Abbreviations:

  • SSRI: Selective Serotonin Reuptake Inhibitor

  • SPARI: Serotonin Partial Agonist and Reuptake Inhibitor

  • SNRI: Serotonin Norepinephrine Reuptake Inhibitor

  • DNRI: Dopamine Norepinephrine Reuptake Inhibitor

  • MAOI: Monoamine Oxidase Inhibitor

  • 5HT2A: Serotonin 2A Receptor

  • SERT: Serotonin Reuptake Pump

Unified Drug Interactions Chart

Drug Class

Psychedelic Class

Interaction Notes

Recommendations

SSRIs (e.g., Paroxetine, Sertraline)

Phenethylamines (MDMA, Mescaline)

Drastically reduced effects due to blocked serotonin reuptake pump.

Taper 2 weeks prior (6 weeks for fluoxetine).

Tryptamines (Psilocybin, LSD)

Potential blunted effects due to receptor downregulation; psilocybin may be less affected.

Taper 2 weeks prior (6 weeks for fluoxetine).

MAOI-containing (Ayahuasca, Syrian Rue)

High risk of serotonin syndrome. Strictly contraindicated.

Avoid combination.

Ketamine

Found effective with or without antidepressants.

No taper required.

Ibogaine

Risk of QTc prolongation, arrhythmias. Some SSRIs inhibit liver enzymes, increasing ibogaine concentration.

Taper 2 weeks prior.

SPARI (e.g., Vilazodone, Vortioxetine)

Phenethylamines

Similar to SSRIs, reduced effects of MDMA.

Taper 2 weeks prior.

Tryptamines

Blunted effects possible.

Taper 2 weeks prior.

MAOI-containing

Risk of serotonin syndrome. Contraindicated.

Avoid combination.

SNRIs (e.g., Venlafaxine, Duloxetine)

Phenethylamines

Similar to SSRIs; reduced MDMA effects.

Taper 2 weeks prior.

Tryptamines

Blunted effects likely.

Taper 2 weeks prior.

MAOI-containing

High risk of serotonin syndrome.

Avoid combination.

Ibogaine

Increased risk of cardiotoxicity.

Taper 2 weeks prior.

DNRI (e.g., Bupropion)

Phenethylamines

Increased MDMA effects; higher seizure risk.

Reduce MDMA dose by 25% or taper bupropion.

Tryptamines

Loss of effect not predicted.

Taper based on goals.

MAOI-containing

Serotonin syndrome unlikely.

Taper 2 weeks prior.

Ibogaine

May increase ibogaine concentration; seizure risk.

Taper 2 weeks prior.

Tricyclic Antidepressants (TCA)

Phenethylamines

Reduced MDMA effects.

Taper 2 weeks prior.

Tryptamines

Intensified LSD effects reported.

Taper 2 weeks prior.

MAOI-containing

High serotonin syndrome risk (especially clomipramine).

Avoid combination.

Trazodone

Phenethylamines

Reduced psychedelic effects at low doses.

Taper 5 days prior.

MAOI-containing

Risk of toxicity.

Taper 1 week prior.

Buspirone

Tryptamines

Blunted effects due to competitive inhibition.

Taper 5 days prior.

MAOI-containing

Low serotonin syndrome risk.

Taper 5 days prior.

MAOI-A (e.g., Phenelzine)

All Psychedelics

High risk of serotonin syndrome, hypertensive crisis.

Taper 2 weeks prior.

Intensified experiences or cardiovascular collapse.

Avoid combination.

MAOI-B (e.g., Selegiline)

Phenethylamines

Intensified MDMA effects; serotonin syndrome risk.

Taper 2 weeks prior if ≥9mg/day.

Tryptamines

Likely low risk with psilocybin, LSD.

Taper 2 weeks prior if ≥9mg/day.

Atypical Antipsychotics(e.g., Aripiprazole, Quetiapine)

All Psychedelics

Potential to blunt psychedelic effects or cause unpredictable interactions.

Avoid combination or consult healthcare provider.

Mood Stabilizers (e.g., Lithium, Valproate)

Phenethylamines/Tryptamines

Lithium poses significant risks (e.g., seizures, serotonin syndrome).

Avoid combination.

Benzodiazepines (e.g., Diazepam, Alprazolam)

All Psychedelics

Can reduce or mitigate psychedelic effects. Often used to manage challenging experiences.

Use with caution for acute situations.

Stimulants (e.g., Methylphenidate, Amphetamine salts)

All Psychedelics

May increase risk of overstimulation or cardiovascular events.

Avoid combination or use with caution.

Opioids (e.g., Morphine, Buprenorphine)

All Psychedelics

Interactions less studied; altered psychedelic experience possible.

Avoid combination without medical supervision.

Anticonvulsants (e.g., Phenytoin, Carbamazepine)

All Psychedelics

Potential altered metabolism and efficacy of psychedelics.

Use with caution or avoid.

Over-the-Counter Medications (e.g., Diphenhydramine, DXM)

All Psychedelics

DXM may cause dangerous serotonin-related interactions.

Avoid combination.

Special Notes:

  • Ketamine: Studied for safe use with antidepressants. The manufacturer recommends combining with oral antidepressants for esketamine therapy.

Ibogaine: CYP2D6 inhibitors (e.g., fluoxetine, bupropion) can double ibogaine concentrations, increasing toxicity risk.

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